Proteins and Drug Design
Oral Contributions
Design of Potent Selective Zinc-Mediated Serine Protease Inhibitors
B.A. Katz, J.M. Clark, J.S. Finer-Moore, T.E. Jenkins, C.R. Johnson, M.J. Ross, C. Luong, W.R. Moore, R. Stroud
Crystal Structures of the Catalytic Domain of HIV-1 Integrase Free and Complexed with its Metal Cofactor: High Similarity of the Active Site with Other Viral Integrases
S. Maignan, J.P. Guilloteau, Qing Zhou-Liu, C. Clement-Mella, V. Mikol
Drug Design and Resistance Mutants in HIV Reverse Transcriptase
D. Stammers
Cell Cycle Inhibition and Drug Design: Crystal Structures of cdk2-inhibitor Complexes
M. Noble,
N. Brown, J. Endicott, L. Johnson, A. Lawrie, J. Tucker, P. Tunnah, A. Calvert, N. Curtin, B. Golding, R. Griffin, D. Newell
Crystal Structure of the Biosenzor Glucose Dehydrogenase
A. Oubrie, H. Rozeboom, K. Kalk, B. Dijkstra
Prolyl oligopeptidase: a beta-propellor regulates cytosolic proteolysis
V. Fülöp
Controlling insulin bioavailability by crystal contact engineering
R. Hilgenfeld, T. Sicker, M. Dörschug, R. Obermeier, K. Geisen, G. Seipke, H. Berchtold
Posters
Structural Studies of Eye-Lense Crystallins.
A.K. Basak, G. Wright, C. Slingsby
Non-Proline CIS Peptide Bonds in Proteins
M.S. Weiss, A. Jabs, R. Hilgenfeld
Neutron Crystallographic Evidence of Lipase/Colipase Complex Activation by a Micelle
J. Hermoso, D. Pignol, S. Penel, M. Roth, C. Chapus, J.C. Fontecilla-Camps
Crystal Structures of Some Prolyl-Oligopeptidase - Inhibitor Complexes
V. Harmat, Zs. Böcskei, V. Fülöp, K. Kánai, G. Náray-Szabó, I. Hermecz, L. Polgár, P. Arányi
Contribution of Rnase Sa Complexes to Protein-Protein/Nucleic Acid Recognition
L. Urbanikova, J. Sevcik
Structural parameters for Proteins Derived from the Atomic Resolution (1.09A) Structure of Designed Variant of the ColE1 Rop Protein
M. Vlassi, M. Kokkinidis
Structure of the Glycosylated Plant Aspartic Proteinase Cardosin A, to 1.72 A Resolution
I. Bento, C. Frazao, R. Coelho, J. Costa, C. Faro, P. Verissimo, E. Pires, J. Cooper, Z. Dauter, K. Wilson, M.A. Carrondo
CAMM of Anticancer Drugs
K. Huml, V. ubr, K. Ulbrich
Structure-Function Studies of Human Ceruloplasmin
V. Zaitsev, I. Zaitseva, G. Card, P. Lindley
Structure of Chitinase from Jack Bean
M. Hahn, M. Hennig, B. Schlesier, W. Höhne
Protein Tiration in the Crystal State
R. Berisio, V.S. Lamzin, F. Sica, K.S. Wilson, A. Zagari, L. Mazzarella
Substrate Complexes of the free radical enzyme Galactose oxidase
E. Vinecombe, S.E.V. Philips
The Crystal Structure of Human Glutathione Reductase Inhibited by Ajoene
S. Bonse, H. Gallwitz, A. Martinez, I. Schlichting, R.L. Krauth-Siegel
A Five-Residue Deletion Alters the Folding and Increases Drastically the Stability of ROP
M. Kokkinidis, G. Cesareni, H.-J. Hinz, Y. Papanikolau, M. Vlassi
Structural Studies of Penicillin binding proteins
E. Gordon, N. Mouz, E. Duee, O. Dideberg
The structure of three inhibitors in complex with HIV-1 protease reveals the importance of structural waters
H.O. Andersson, J. Hulten, S. Löwgren, N.M. Bonham, W. Schaal, A. Karlen, A. Hallberg, T. Unge
Structural studies of purple acid phosphatase from rat bone.
Jia Jia, E. Johansson, H. Kaija, P. Vihko, G. Schneider, Y. Lindqvist
The Structure of Pore-Forming Proteins in Prokaryotes and Eurokaryotes
K. Zeth, J. Diez, M. Dolder, V. Adams, K. Diederichs, W. Welte, T. Wallimann, H. Engelhardt
Crystal Structure of Pneumocystis Carinii Dihydrofolate Reductase Cofactor Complex with Tab, a Potent, PC-Selective Antifolate
N. Galitsky, V. Cody, D. rak, J.R. Luft, W. Pangborn, S.F. Queener, M.F.G. Stevens, C. Laughton, D. Chan
Crystal Structure of S58A Mutant of E. coli L-Asparaginase II
M. Kozak, M. Jaskolski
Studies of Papain in Complex with Epoxysuccinyl-peptide Inhibitor
M. Kozak, E. Jankowska, J. Ciarkowski, Z. Grzonka, M. Jaskolski
The crystal structure of beta-ketoacyl [ACP] synthase I from Escherichia coli
J.G. Olsen, A. Kadziola, P. von Wettstein-Knowles, S. Larsen
Crystallographic Studies of Mammaian Pentraxins
D. Thompson, M.B. Pepys, S.P. Wood
The use of X-ray crystal structures in the design of novel, potent thrombin inhibitors.
A. Cleasby, H. Jhotti, S. Patel, A. Wonacott, M. Weir
High Resolution Crystal Structure of a Histamine-Binding Rhipicephalus Appendiculatus
P. Adams, G.C. Paesen, K. Harlso, P.A. Nutta, D.I. Stuart
Crystals of FAB+hCG complex and fabs.
M.A. Dingwall, N.W. Isaacs
Anti-Retroviral Drug Design Based on Structure Analysis of Proteases
J. Hasek, J. Dohnalek, J. Duskova, J. Konvalinka, M. Hradilek, M. Soucek, J. Sedlacek, J. Brynda, E. Buchtelova